Initial Solvent Screening of Carbamazepine, Cimetidine, and Phenylbutazone: Part 1 of 2 - Pharmaceutical Technology

Latest Issue
PharmTech

Latest Issue
PharmTech Europe

Initial Solvent Screening of Carbamazepine, Cimetidine, and Phenylbutazone: Part 1 of 2
The authors describe the importance of a rapid and an abbreviated screening strategy by initial solvent screening in 20-mL scintillation vials.


Pharmaceutical Technology
Volume 33, Issue 5, pp. 62-72

References

1. Y. Kawashima and C.E. Capes, "An Experimental Study of the Kinetics of Spherical Agglomeration in a Stirred Vessel," Powder Technol. 10 (1–2), 85–92 (1974).

2. Y. Kawashima and C.E. Capes, "Further Studies of the Kinetics of Spherical Agglomeration in a Stirred Vessel," Powder Technol. 13 (2), 279–288 (1976).

3. Y. Kawashima, M. Okumura, and H. Takenaka, "Spherical Crystallization: Direct Spherical Agglomeration of Salicylic Acid Crystals During Crystallization," Science 216 (4550), 1127–1128 (1982).

4. Y. Kawashima et al., "Preparation of Spherically Agglomerated Crystals of Aminophylline," J. Pharm. Sci. 73 (10), 1407–1409 (1984).

5. Y. Kawashima, M. Okumura, and H. Takenaka, "The Effects of Temperature on the Spherical Crystallization of Salicylic Acid," Powder Technol. 39 (1), 41–47 (1984).

6. Y. Kawashima et al., "Preparations of Agglomerated Crystals of Polymorphic Mixtures and a New Complex of Indomethacin-Epirizole by the Spherical Crystallization Technique," J. Pharm. Sci. 74 (11), 1152–1156 (1985).

7. A. Sano et al., "Particle Design of Tolbutamide by the Spherical Crystallization Technique II: Factors Causing Polymorphism of Tolbutamide Spherical Agglomerates," Chem. Pharm. Bull. 37 (8), 2183–2187 (1989).

8. Y. Kawashima et al., "Characterization of Polymorphs of Tranilast Anhydrate and Tranilast Monohydrate When Crystallized by Two Solvent Change Spherical Crystallization Techniques," J. Pharm. Sci. 80 (5), 472–478 (1991).

9. K. Morishima et al., "Micromeritic Characteristics and Agglomeration Mechanisms in the Spherical Crystallization of Bucillamine by the Spherical Agglomeration and the Emulsion Solvent Diffusion Methods," Powder Technol. 76 (1), 57–64 (1993).

10. Y. Kawashima et al., "Improvements in Flowability and Compressibility of Pharmaceutical Crystals for Direct Tabletting by Spherical Crystallization with a Two-Solvent System," Powder Technol. 78 (2), 151–157 (1994).

11. K. Morishima et al., "Tabletting Properties of Bucillamine Agglomerates Prepared by the Spherical Crystallization Technique," Int. J. Pharm. 105 (11), 11–18 (1994).

12. A.M. Garcia and E.S. Ghaly, "Preliminary Spherical Agglomerates of Water Soluble Drug Using Natural Polymer and Cross-Linking Technique," J. Control. Release 40 (3), 179–186 (1996).

13. A.H.L. Chow and M.W.M. Leung, "A Study of the Mechanisms of Wet Spherical Agglomeration of Pharmaceutical Powders," Drug Dev. Ind. Pharm. 22 (4), 357–371 (1996).

14. U. Teipel, T. Heintz, and H.H. Krause, "Crystallization of Spherical Ammonium Dinitramide (ADN) Particles," Propellants, Explosives, Pyrotechnics 25 (2), 81–85 (2000).

15. P. Szabó-Révész et al., "Development of Spherical Crystal Agglomerates of an Aspartic Acid Salt for Direct Tablet Making," Powder Technol. 114 (1), 118–124 (2001).

16. A.R. Paradkar et al., "Spherical Crystallization of Celecoxib," Drug Dev. Ind. Pharm. 28 (10), 1213–1220 (2002).

17. P. Szabó -Révész et al., "Crystal Growth of Drug Materials by Spherical Crystallization," J. Cryst. Growth 237–239 (part 3), 2240–2245 (2002).

18. Y. Kawashima et al., "Improved Flowability and Compactibility of Spherically Agglomerated Crystals of Ascorbic Acid for Direct Tableting Designed by Spherical Crystallization Process," Powder Technol. 130 (1), 283–289 (2003).

19. A.P. Pawar et al., "Crystallo-co-agglomeration: A Novel Technique to Obtain Ibuprofen-Paracetamol Agglomerates," AAPS Pharm. Sci. Tech., 5 (3), Article 44 (2004).

20. S. Bhadra et al., "Spherical Crystallization of Mefenamic Acid," Pharm. Technol. 28 (2), 66–76 (2004).

21. M. Maghsoodi et al., "Improved Compaction and Packing Properties of Naproxen Agglomerated Crystals Obtained by Spherical Crystallization Technique," Drug Dev. Ind. Pharm. 33 (11), 1216–1224 (2007).

22. J. Katta and ĺ.C. Rasmuson, "Spherical Crystallization of Benzoic Acid," Int. J. Pharm. 348 (1–2), 61–69 (2008).

23. X. Liu et al., "Single-Crystal-like Materials by the Self-Assembly of Cube-Shaped Lead Zirconate Titanate (PZT) Microcrystals," Langmuir 21 (8), 3207–3212 (2005).

24. A.S. Utada et al., "Monodisperse Double Emulsions Generated from a Microcapillary Device," Science 308 (5721), 537–541 (2005).

25. S. Gupta and S.P. Moulik, "Biocompatible Microemulsions and Their Prospective Uses in Drug Delivery," J. Pharm. Sci. 97 (1), 22–45 (2008).

26. K. Ujiiye-Ishii et al., "Methodological Features of the Emulsion and Reprecipitation Methods for Organic Nanocrystal Fabrication," Cryst. Growth Des. 8 (2), 369–371 (2008).

27. T. Lee and S.T. Hung, "Cocktail-Solvent Screening to Enhance Solubility, Increase Crystal Yield, and Induce Polymorphs," Pharm. Technol. 32 (1), 76–95 (2008).

28. T. Lee, C.S. Kuo, and Y.H. Chen, "Solubility, Polymorphism, Crystallinity, and Crystal Habit of Acetaminophen and Ibuprofen," Pharm. Technol. 30 (10), 72–92 (2006).

29. T. Lee, Y.H. Chen, and C.W. Zhang, "Solubility, Polymorphism, Crystallinity, Crystal Habit, and Drying Scheme of (R,S)-(±)-Sodium Ibuprofen Dihydrate," Pharm. Technol. 31 (6), 72–87 (2007).

30. T. Lee and M.S. Lin, "Sublimation Point Depression of Tris(8-hydroxyquinoline)aluminum(III) (Alq3) by Crystal Engineering," Cryst. Growth Des. 7 (9), 1803–1810 (2007).

31. J. Alsenz and M. Kansy, "High Throughput Solubility Measurement in Drug Discovery and Development," Adv. Drug Deliv. Rev. 59 (7), 546–567 (2007).


ADVERTISEMENT

blog comments powered by Disqus
LCGC E-mail Newsletters

Subscribe: Click to learn more about the newsletter
| Weekly
| Monthly
|Monthly
| Weekly

Survey
What role should the US government play in the current Ebola outbreak?
Finance development of drugs to treat/prevent disease.
Oversee medical treatment of patients in the US.
Provide treatment for patients globally.
All of the above.
No government involvement in patient treatment or drug development.
Finance development of drugs to treat/prevent disease.
27%
Oversee medical treatment of patients in the US.
14%
Provide treatment for patients globally.
8%
All of the above.
41%
No government involvement in patient treatment or drug development.
11%
Jim Miller Outsourcing Outlook Jim MillerCMO Industry Thins Out
Cynthia Challener, PhD Ingredients Insider Cynthia ChallenerFluorination Remains Key Challenge in API Synthesis
Marilyn E. Morris Guest EditorialMarilyn E. MorrisBolstering Graduate Education and Research Programs
Jill Wechsler Regulatory Watch Jill Wechsler Biopharma Manufacturers Respond to Ebola Crisis
Sean Milmo European Regulatory WatchSean MilmoHarmonizing Marketing Approval of Generic Drugs in Europe
FDA Reorganization to Promote Drug Quality
FDA Readies Quality Metrics Measures
New FDA Team to Spur Modern Drug Manufacturing
From Generics to Supergenerics
CMOs and the Track-and-Trace Race: Are You Engaged Yet?
Source: Pharmaceutical Technology,
Click here