Initial Solvent Screening of Carbamazepine, Cimetidine, and Phenylbutazone: Part 1 of 2 - Pharmaceutical Technology

Latest Issue
PharmTech

Latest Issue
PharmTech Europe

Initial Solvent Screening of Carbamazepine, Cimetidine, and Phenylbutazone: Part 1 of 2
The authors describe the importance of a rapid and an abbreviated screening strategy by initial solvent screening in 20-mL scintillation vials.


Pharmaceutical Technology
Volume 33, Issue 5, pp. 62-72

References

1. Y. Kawashima and C.E. Capes, "An Experimental Study of the Kinetics of Spherical Agglomeration in a Stirred Vessel," Powder Technol. 10 (1–2), 85–92 (1974).

2. Y. Kawashima and C.E. Capes, "Further Studies of the Kinetics of Spherical Agglomeration in a Stirred Vessel," Powder Technol. 13 (2), 279–288 (1976).

3. Y. Kawashima, M. Okumura, and H. Takenaka, "Spherical Crystallization: Direct Spherical Agglomeration of Salicylic Acid Crystals During Crystallization," Science 216 (4550), 1127–1128 (1982).

4. Y. Kawashima et al., "Preparation of Spherically Agglomerated Crystals of Aminophylline," J. Pharm. Sci. 73 (10), 1407–1409 (1984).

5. Y. Kawashima, M. Okumura, and H. Takenaka, "The Effects of Temperature on the Spherical Crystallization of Salicylic Acid," Powder Technol. 39 (1), 41–47 (1984).

6. Y. Kawashima et al., "Preparations of Agglomerated Crystals of Polymorphic Mixtures and a New Complex of Indomethacin-Epirizole by the Spherical Crystallization Technique," J. Pharm. Sci. 74 (11), 1152–1156 (1985).

7. A. Sano et al., "Particle Design of Tolbutamide by the Spherical Crystallization Technique II: Factors Causing Polymorphism of Tolbutamide Spherical Agglomerates," Chem. Pharm. Bull. 37 (8), 2183–2187 (1989).

8. Y. Kawashima et al., "Characterization of Polymorphs of Tranilast Anhydrate and Tranilast Monohydrate When Crystallized by Two Solvent Change Spherical Crystallization Techniques," J. Pharm. Sci. 80 (5), 472–478 (1991).

9. K. Morishima et al., "Micromeritic Characteristics and Agglomeration Mechanisms in the Spherical Crystallization of Bucillamine by the Spherical Agglomeration and the Emulsion Solvent Diffusion Methods," Powder Technol. 76 (1), 57–64 (1993).

10. Y. Kawashima et al., "Improvements in Flowability and Compressibility of Pharmaceutical Crystals for Direct Tabletting by Spherical Crystallization with a Two-Solvent System," Powder Technol. 78 (2), 151–157 (1994).

11. K. Morishima et al., "Tabletting Properties of Bucillamine Agglomerates Prepared by the Spherical Crystallization Technique," Int. J. Pharm. 105 (11), 11–18 (1994).

12. A.M. Garcia and E.S. Ghaly, "Preliminary Spherical Agglomerates of Water Soluble Drug Using Natural Polymer and Cross-Linking Technique," J. Control. Release 40 (3), 179–186 (1996).

13. A.H.L. Chow and M.W.M. Leung, "A Study of the Mechanisms of Wet Spherical Agglomeration of Pharmaceutical Powders," Drug Dev. Ind. Pharm. 22 (4), 357–371 (1996).

14. U. Teipel, T. Heintz, and H.H. Krause, "Crystallization of Spherical Ammonium Dinitramide (ADN) Particles," Propellants, Explosives, Pyrotechnics 25 (2), 81–85 (2000).

15. P. Szabó-Révész et al., "Development of Spherical Crystal Agglomerates of an Aspartic Acid Salt for Direct Tablet Making," Powder Technol. 114 (1), 118–124 (2001).

16. A.R. Paradkar et al., "Spherical Crystallization of Celecoxib," Drug Dev. Ind. Pharm. 28 (10), 1213–1220 (2002).

17. P. Szabó -Révész et al., "Crystal Growth of Drug Materials by Spherical Crystallization," J. Cryst. Growth 237–239 (part 3), 2240–2245 (2002).

18. Y. Kawashima et al., "Improved Flowability and Compactibility of Spherically Agglomerated Crystals of Ascorbic Acid for Direct Tableting Designed by Spherical Crystallization Process," Powder Technol. 130 (1), 283–289 (2003).

19. A.P. Pawar et al., "Crystallo-co-agglomeration: A Novel Technique to Obtain Ibuprofen-Paracetamol Agglomerates," AAPS Pharm. Sci. Tech., 5 (3), Article 44 (2004).

20. S. Bhadra et al., "Spherical Crystallization of Mefenamic Acid," Pharm. Technol. 28 (2), 66–76 (2004).

21. M. Maghsoodi et al., "Improved Compaction and Packing Properties of Naproxen Agglomerated Crystals Obtained by Spherical Crystallization Technique," Drug Dev. Ind. Pharm. 33 (11), 1216–1224 (2007).

22. J. Katta and å.C. Rasmuson, "Spherical Crystallization of Benzoic Acid," Int. J. Pharm. 348 (1–2), 61–69 (2008).

23. X. Liu et al., "Single-Crystal-like Materials by the Self-Assembly of Cube-Shaped Lead Zirconate Titanate (PZT) Microcrystals," Langmuir 21 (8), 3207–3212 (2005).

24. A.S. Utada et al., "Monodisperse Double Emulsions Generated from a Microcapillary Device," Science 308 (5721), 537–541 (2005).

25. S. Gupta and S.P. Moulik, "Biocompatible Microemulsions and Their Prospective Uses in Drug Delivery," J. Pharm. Sci. 97 (1), 22–45 (2008).

26. K. Ujiiye-Ishii et al., "Methodological Features of the Emulsion and Reprecipitation Methods for Organic Nanocrystal Fabrication," Cryst. Growth Des. 8 (2), 369–371 (2008).

27. T. Lee and S.T. Hung, "Cocktail-Solvent Screening to Enhance Solubility, Increase Crystal Yield, and Induce Polymorphs," Pharm. Technol. 32 (1), 76–95 (2008).

28. T. Lee, C.S. Kuo, and Y.H. Chen, "Solubility, Polymorphism, Crystallinity, and Crystal Habit of Acetaminophen and Ibuprofen," Pharm. Technol. 30 (10), 72–92 (2006).

29. T. Lee, Y.H. Chen, and C.W. Zhang, "Solubility, Polymorphism, Crystallinity, Crystal Habit, and Drying Scheme of (R,S)-(±)-Sodium Ibuprofen Dihydrate," Pharm. Technol. 31 (6), 72–87 (2007).

30. T. Lee and M.S. Lin, "Sublimation Point Depression of Tris(8-hydroxyquinoline)aluminum(III) (Alq3) by Crystal Engineering," Cryst. Growth Des. 7 (9), 1803–1810 (2007).

31. J. Alsenz and M. Kansy, "High Throughput Solubility Measurement in Drug Discovery and Development," Adv. Drug Deliv. Rev. 59 (7), 546–567 (2007).


ADVERTISEMENT

blog comments powered by Disqus
LCGC E-mail Newsletters

Subscribe: Click to learn more about the newsletter
| Weekly
| Monthly
|Monthly
| Weekly

Survey
How does your company apply quality-by-design (QbD) principles to manufacturing processes?
To all processes for both new and legacy products
To all process for new products only
To select process for new products only
To select processes for both new and legacy products
Do not use QbD
To all processes for both new and legacy products
21%
To all process for new products only
13%
To select process for new products only
26%
To select processes for both new and legacy products
21%
Do not use QbD
21%
View Results
UPCOMING CONFERENCES

Programs for Investigational and Pre-Launch Drugs
Philadelphia, PA
July 17-18, 2013
Request Brochure

Strategic Pipeline Planning & Portfolio Valuation
Philadelphia, PA
August 13-14, 2013
Request Brochure

MES 2013 - Forum on Manufacturing Execution Systems
Philadelphia, PA
August 14-15, 2013
Request Brochure

Mobile Innovation for the Life Sciences Industry
Philadelphia, PA
August 20-21, 2013
Request Brochure

See All Conferences >>

Eric Langer Outsourcing Outlook Eric LangerOutsourcing's Modest Role as a Cost-Containment Strategy
Patricia Van Arnum Ingredients Insider Patricia Van ArnumIntellectual Property Battles in Solid-State Chemistry
Nathan Jessop Industry Insider Nathan Jessop Campaign Against Counterfeit Drugs Continues
Lynn Torbeck Statistical Solutions Lynn D. TorbeckCompositing Samples and the Risk to Product Quality
 More
Global Biosimilars Market to Reach $2.445 Billion in 2013
Adapting to Change
AstraZeneca and Exco InTouch Collaborate to Augment Current COPD Pathways
Overcoming the Challenges in Biopharmaceutical Stability Testing
PhRMA Dismayed by Special 301 Report
FindPharma Custom Search
Source: Pharmaceutical Technology,
Click here